Class information for:
Level 1: FLUORESCENT LIGANDS//1012 S//ALEXA FLUOR R 647

Basic class information

Class id #P Avg. number of
references
Database coverage
of references
32378 140 37.1 67%



Bar chart of Publication_year

Last years might be incomplete

Hierarchy of classes

The table includes all classes above and classes immediately below the current class.



Cluster id Level Cluster label #P
0 4 BIOCHEMISTRY & MOLECULAR BIOLOGY//CELL BIOLOGY//ONCOLOGY 4064930
405 3       BACTERIORHODOPSIN//G PROTEIN COUPLED RECEPTOR//G PROTEIN 29641
705 2             G PROTEIN COUPLED RECEPTOR//GPCR//RHODOPSIN 12950
32378 1                   FLUORESCENT LIGANDS//1012 S//ALEXA FLUOR R 647 140

Terms with highest relevance score



rank Term termType Chi square Shr. of publ. in
class containing
term
Class's shr. of
term's tot. occurrences
#P with
term in
class
1 FLUORESCENT LIGANDS authKW 1090545 7% 50% 10
2 1012 S authKW 218111 1% 100% 1
3 ALEXA FLUOR R 647 authKW 218111 1% 100% 1
4 ANTHROYLCHOLINE BROMIDE authKW 218111 1% 100% 1
5 AVIDIN BIOTIN BINDING ASSAY authKW 218111 1% 100% 1
6 BIOTIN 1012S CONJUGATE authKW 218111 1% 100% 1
7 BIOTIN AND FLUORESCENCE LABELING authKW 218111 1% 100% 1
8 BODIPY TMR CGP authKW 218111 1% 100% 1
9 BRITISH PHARMACOLOGICAL SOCIETY 75TH ANNIVERSARY authKW 218111 1% 100% 1
10 CHEMOKINE AND CHOLECYSTOKININ RECEPTORS authKW 218111 1% 100% 1

Web of Science journal categories



Rank Term Chi square Shr. of publ. in
class containing
term
Class's shr. of
term's tot. occurrences
#P with
term in
class
1 Chemistry, Medicinal 1219 28% 0% 39
2 Pharmacology & Pharmacy 435 34% 0% 47
3 Chemistry, Analytical 116 14% 0% 19
4 Biochemistry & Molecular Biology 83 24% 0% 33
5 Chemistry, Organic 34 9% 0% 12
6 Cell Biology 29 9% 0% 13
7 Biochemical Research Methods 21 5% 0% 7
8 Biophysics 16 5% 0% 7
9 Neurosciences 15 9% 0% 12
10 Biology 8 3% 0% 4

Address terms



Rank Term Chi square Shr. of publ. in
class containing
term
Class's shr. of
term's tot. occurrences
#P with
term in
class
1 CISBIO BIOASSAYS 218111 1% 100% 1
2 ESBSIFR 85 218111 1% 100% 1
3 INNOVAT THER EUT MEDALISUMR7200 218111 1% 100% 1
4 NEUROPEPTIDES CENT REGULAT HYDR CARDIOVASC 218111 1% 100% 1
5 PCBISFMTSUMS 3286 218111 1% 100% 1
6 UDS EX MEDALIS PHARMUMR 7200 218111 1% 100% 1
7 UDS PHARMUMR 7213 218111 1% 100% 1
8 UMR 7081ULPIFR 85 218111 1% 100% 1
9 UMR INSERM U1050 7241 218111 1% 100% 1
10 CELL SIGNALLING 143892 13% 4% 18

Journals



Rank Term Chi square Shr. of publ. in
class containing
term
Class's shr. of
term's tot. occurrences
#P with
term in
class
1 JOURNAL OF RECEPTOR RESEARCH 1498 1% 0% 2
2 ANALYTICAL LETTERS 1172 4% 0% 6
3 JOURNAL OF MEDICINAL CHEMISTRY 1007 7% 0% 10
4 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 856 7% 0% 10
5 CELL COMMUNICATION AND SIGNALING 578 1% 0% 1
6 MOLECULAR PHARMACOLOGY 552 4% 0% 5
7 JOURNAL OF BIOMOLECULAR SCREENING 506 1% 0% 2
8 REVISTA ESPANOLA DE LAS ENFERMEDADES DEL APARATO DIGESTIVO 452 1% 0% 1
9 CURRENT MEDICINAL CHEMISTRY 441 2% 0% 3
10 BRITISH JOURNAL OF PHARMACOLOGY 435 4% 0% 6

Author Key Words



Rank Term Chi square Shr. of publ. in
class containing
term
Class's shr. of
term's tot. occurrences
#P with
term in
class
LCSH search Wikipedia search
1 FLUORESCENT LIGANDS 1090545 7% 50% 10 Search FLUORESCENT+LIGANDS Search FLUORESCENT+LIGANDS
2 1012 S 218111 1% 100% 1 Search 1012+S Search 1012+S
3 ALEXA FLUOR R 647 218111 1% 100% 1 Search ALEXA+FLUOR+R+647 Search ALEXA+FLUOR+R+647
4 ANTHROYLCHOLINE BROMIDE 218111 1% 100% 1 Search ANTHROYLCHOLINE+BROMIDE Search ANTHROYLCHOLINE+BROMIDE
5 AVIDIN BIOTIN BINDING ASSAY 218111 1% 100% 1 Search AVIDIN+BIOTIN+BINDING+ASSAY Search AVIDIN+BIOTIN+BINDING+ASSAY
6 BIOTIN 1012S CONJUGATE 218111 1% 100% 1 Search BIOTIN+1012S+CONJUGATE Search BIOTIN+1012S+CONJUGATE
7 BIOTIN AND FLUORESCENCE LABELING 218111 1% 100% 1 Search BIOTIN+AND+FLUORESCENCE+LABELING Search BIOTIN+AND+FLUORESCENCE+LABELING
8 BODIPY TMR CGP 218111 1% 100% 1 Search BODIPY+TMR+CGP Search BODIPY+TMR+CGP
9 BRITISH PHARMACOLOGICAL SOCIETY 75TH ANNIVERSARY 218111 1% 100% 1 Search BRITISH+PHARMACOLOGICAL+SOCIETY+75TH+ANNIVERSARY Search BRITISH+PHARMACOLOGICAL+SOCIETY+75TH+ANNIVERSARY
10 CHEMOKINE AND CHOLECYSTOKININ RECEPTORS 218111 1% 100% 1 Search CHEMOKINE+AND+CHOLECYSTOKININ+RECEPTORS Search CHEMOKINE+AND+CHOLECYSTOKININ+RECEPTORS

Core articles

The table includes core articles in the class. The following variables is taken into account for the relevance score of an article in a cluster c:
(1) Number of references referring to publications in the class.
(2) Share of total number of active references referring to publications in the class.
(3) Age of the article. New articles get higher score than old articles.
(4) Citation rate, normalized to year.



Rank Reference # ref.
in cl.
Shr. of ref. in
cl.
Citations
1 KOZMA, E , JAYASEKARA, PS , SQUARCIALUPI, L , PAOLETTA, S , MORO, S , FEDERICO, S , SPALLUTO, G , JACOBSON, KA , (2013) FLUORESCENT LIGANDS FOR ADENOSINE RECEPTORS.BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. VOL. 23. ISSUE 1. P. 26 -36 21 58% 11
2 KUDER, K , KIEC-KONONOWICZ, K , (2008) FLUORESCENT GPCR LIGANDS AS NEW TOOLS IN PHARMACOLOGY.CURRENT MEDICINAL CHEMISTRY. VOL. 15. ISSUE 21. P. 2132-2143 18 56% 23
3 SRIDHARAN, R , ZUBER, J , CONNELLY, SM , MATHEW, E , DUMONT, ME , (2014) FLUORESCENT APPROACHES FOR UNDERSTANDING INTERACTIONS OF LIGANDS WITH G PROTEIN COUPLED RECEPTORS.BIOCHIMICA ET BIOPHYSICA ACTA-BIOMEMBRANES. VOL. 1838. ISSUE 1. P. 15-33 45 14% 23
4 STODDART, LA , KILPATRICK, LE , BRIDDON, SJ , HILL, SJ , (2015) PROBING THE PHARMACOLOGY OF G PROTEIN-COUPLED RECEPTORS WITH FLUORESCENT LIGANDS.NEUROPHARMACOLOGY. VOL. 98. ISSUE . P. 48 -57 23 30% 4
5 JANSSEN, MJ , ENSING, K , DE ZEEUW, RA , (2001) A FLUORESCENT RECEPTOR ASSAY FOR BENZODIAZEPINES USING COUMARIN LABELED DESETHYLFLUMAZENIL AS LIGAND.ANALYTICAL CHEMISTRY. VOL. 73. ISSUE 13. P. 3168-3173 11 92% 5
6 VERNALL, AJ , HILL, SJ , KELLAM, B , (2014) THE EVOLVING SMALL-MOLECULE FLUORESCENT-CONJUGATE TOOLBOX FOR CLASS A GPCRS.BRITISH JOURNAL OF PHARMACOLOGY. VOL. 171. ISSUE 5. P. 1073-1084 16 36% 10
7 KUDER, KJ , KIEC-KONONOWICZ, K , (2014) FLUORESCENT GPCR LIGANDS AS NEW TOOLS IN PHARMACOLOGY-UPDATE, YEARS 2008-EARLY 2014.CURRENT MEDICINAL CHEMISTRY. VOL. 21. ISSUE 34. P. 3962 -3975 16 37% 2
8 STODDART, LA , WHITE, CW , NGUYEN, K , HILL, SJ , PFLEGER, KDG , (2016) FLUORESCENCE- AND BIOLUMINESCENCE-BASED APPROACHES TO STUDY GPCR LIGAND BINDING.BRITISH JOURNAL OF PHARMACOLOGY. VOL. 173. ISSUE 20. P. 3028 -3037 16 30% 2
9 JANSSEN, MJ , HULST, R , KELLOGG, RM , HENDRIKS, MMWB , ENSING, K , DE ZEEUW, RA , (2000) FLUORESCENT-LABELED LIGANDS FOR THE BENZODIAZEPINE RECEPTOR - PART 1: SYNTHESIS AND CHARACTERIZATION OF FLUORESCENT-LABELED BENZODIAZEPINES.PHARMAZIE. VOL. 55. ISSUE 1. P. 42-48 10 77% 4
10 CIRUELA, F , FERNANDEZ-DUEHAS, V , JACOBSON, KA , (2015) LIGHTING UP G PROTEIN-COUPLED PURINERGIC RECEPTORS WITH ENGINEERED FLUORESCENT LIGANDS.NEUROPHARMACOLOGY. VOL. 98. ISSUE . P. 58 -67 19 24% 3

Classes with closest relation at Level 1



Rank Class id link
1 9142 RECEPTOR MOSAICS//HETEROMER//RECEPTOR RECEPTOR INTERACTIONS
2 9656 JOURNAL OF BIOMOLECULAR SCREENING//ASSAY AND DRUG DEVELOPMENT TECHNOLOGIES//PHOS TAG
3 3075 MOL RECOGNIT SECT//ADENOSINE RECEPTORS//ADENOSINE RECEPTOR ANTAGONISTS
4 7397 FLUORESCENCE CORRELATION SPECTROSCOPY//SUPRAMOL BIOPHYS//FLUORESCENCE CORRELATION SPECTROSCOPY FCS
5 25076 BIOIMAGING PROBE DEV//SING ORE BIOIMAGING CONSORTIUM//56 CARBOXY RHODAMINE 110
6 10380 XANOMELINE//M 1//ALCURONIUM
7 19599 MOL BIOSENSOR IMAGING//FLUOROGEN ACTIVATING PROTEIN//FLUOROGEN
8 7382 JOURNAL OF CYCLIC NUCLEOTIDE RESEARCH//JOURNAL OF CYCLIC NUCLEOTIDE AND PROTEIN PHOSPHORYLATION RESEARCH//JOURNAL OF RECEPTOR RESEARCH
9 26108 BIOCHEM TECHNOL SCI TECHNOL//GPR35//RESONANT WAVEGUIDE GRATING BIOSENSOR
10 8730 BETA3 ADRENOCEPTOR//BRL 37344//ATYPICAL BETA ADRENOCEPTORS

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